REVIEW Pseudopelletierine oxime, the oxime of 3-tropinone, is a key intermediate in the synthesis of Dolasetron (dolasetron mesilate) a 5-HT3 antagonist.
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Hadley, Michael Stewart; King, Francis David Azabicycloalkyl derivatives and pharmaceutical compositions containing them. Eur. Pat. Appl. (1980), EP 13138 A1 19800709.
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Vernekar, Sanjeev Kumar V.; Hallaq, Hasan Y.; Clarkson, Guy; Thompson, Andrew J.; Silvestri, Linda; Lummis, Sarah C. R.; Lochner, Martin Toward Biophysical Probes for the 5-HT3 Receptor: Structure-Activity Relationship Study of Granisetron Derivatives. Journal of Medicinal Chemistry (2010), 53(5), 2324-2328.
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