REVIEW Inhibits plasma cholinesterase during metabolism. Bambuterol is a racemic phenylethanolamine based long acting beta-adrenoceptor agonist, used in the treatment of asthma; it also is a biscarbamate ester prodrug of the beta 2 adrenergic agonist terbutaline.
Olsson, Otto Agne; Svensson, Leif Ake; Wetterlin, Kjell Ingvar Leopold 1-(Dihydroxyphenyl)-2-aminoethanol derivatives, their compositions and intermediates Eur. Pat. Appl. (1982), EP 43807 A2 19820113.
Svensson LA.Bambuterol- a prodrug-prodrug with built-in hydrolysis brake. Acta Pharm Suec. 1987;24(6):333-41.
Svensson LA.Mechanism of action of bambuterol: a beta-agonist prodrug with sustained lung affinity. Agents Actions Suppl. 1991;34:71-8.
Sitar DS.Clinical pharmacokinetics of bambuterol.Clin Pharmacokinet. 1996 Oct;31(4):246-56.
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